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Synthesis, Characterization, and Antiproliferative Activity Studies of Novel Benzimidazole-Imidazopyridine Hybrids as DNA Groove Binders

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dc.creator Yildiz, Ufuk
dc.creator AKKOÇ, Senem
dc.creator Gercek, Zuhal
dc.creator Sengul, Abdurrahman
dc.creator Coban, Burak
dc.creator Caymaz, Bahar
dc.date 2020-06-30T21:00:00Z
dc.date.accessioned 2020-10-06T09:15:41Z
dc.date.available 2020-10-06T09:15:41Z
dc.identifier 0023a6b5-e3c7-4e77-b264-b0ae836eaefc
dc.identifier 10.1002/slct.202001580
dc.identifier https://avesis.sdu.edu.tr/publication/details/0023a6b5-e3c7-4e77-b264-b0ae836eaefc/oai
dc.identifier.uri http://acikerisim.sdu.edu.tr/xmlui/handle/123456789/51855
dc.description A novel benzimidazole-imidazo[1,2-a]pyridine hybrid; 2-(imidazo[1,2-a]pyridine-8-yl)benzimidazole and its symmetrical bis- derivative 2,2 '-bis-(imidazo[1,2-a]pyridine-8-yl)-1H,1H '-[5,5 ']-bisbenzimidazole were synthesized and characterized. It was found that these two compounds have a strong DNA groove binding and peroxide mediated DNA-cleavage properties. Furthermore, these molecules were screened against three different human cell lines namely HepG2, DLD-1 and MDA-MB-231, and these compounds were found to have high cytotoxic activities.
dc.language eng
dc.rights info:eu-repo/semantics/closedAccess
dc.title Synthesis, Characterization, and Antiproliferative Activity Studies of Novel Benzimidazole-Imidazopyridine Hybrids as DNA Groove Binders
dc.type info:eu-repo/semantics/article


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